SCHEMBL6559766

SCHEMBL6559766

O=C(CO)c1ccc(Cl)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 2/20 0.47
KCNQ2 O43526 2/20 0.47
KCNE1 P15382 2/20 0.47
KCNQ1 P51787 2/20 0.47
KCNQ5 Q9NR82 1/20 0.47
KMO O15229 3/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
TSHR P16473 1/20 0.41
MAOB P27338 3/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
ERCC5 P28715 1/20 0.39
FEN1 P39748 1/20 0.39
HSD11B1 P28845 1/20 0.39
S1PR1 P21453 1/20 0.39
S1PR3 Q99500 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30467135 1.00 KCNQ3 (0.47) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL27503767 0.86 KCNQ3 (0.44) KCNQ3KCNQ2KCNE1KCNQ1KMO
SCHEMBL30025571 0.86 GSK3B (0.53) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL3502522 0.86 KCNQ3 (0.46) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL2630705 0.86 GSK3B (0.53) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL29499477 0.85 GSK3B (0.55) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL13116542 0.85 KCNQ3 (0.45) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL3973133 0.85 GSK3B (0.55) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL18538090 0.85 MAPT (0.54) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5
SCHEMBL2273688 0.83 CES2 (0.61) KCNQ3KCNQ2KCNQ5CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188194-B1 AMINOACRYLIC ACID DERIVATIVES BAYER AG (DE) 1990-07-04 EP claimed
EP-0188194-A2 Aminoacrylic acid derivatives BAYER AG (DE) 1986-07-23 EP claimed
CN-86100221-A AMINOACRYLIC ACID DERIVATIVES 1986-07-16 CN claimed
EP-3494971-B1 SALTS OF ERK INHIBITORS GENENTECH INC (US) 2024-07-24 EP disclosed
CN-111777594-B Method for preparing a medicament 基因泰克公司 2023-06-27 CN disclosed
US-11066389-B2 Process for the manufacturing of medicaments GENENTECH, INC. (US) 2021-07-20 US disclosed
US-11066389-B2 Process for the manufacturing of medicaments GENENTECH, INC. (US) 2021-07-20 US disclosed
US-20200190061-A1 PROCESS FOR THE MANUFACTURING OF MEDICAMENTS GENENTECH, INC. (US) 2020-06-18 US disclosed
US-20200190061-A1 PROCESS FOR THE MANUFACTURING OF MEDICAMENTS GENENTECH, INC. (US) 2020-06-18 US disclosed
US-10611753-B2 Process for the manufacturing of medicaments GENENTECH, INC. (US) 2020-04-07 US disclosed
US-10611753-B2 Process for the manufacturing of medicaments GENENTECH, INC. (US) 2020-04-07 US disclosed
EP-0807629-B1 Sulfonamido substituted chromane derivatives, method for their preparation, their use as medicaments or diagnostic agents aswell as medicaments containing them AVENTIS PHARMA GMBH (DE) 2004-03-03 EP disclosed
US-6191164-B1 POTASSIUM CHANNEL MODULATORS; ANTIULCER AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 2001-02-20 US disclosed
US-6071953-A Sulfonamide-substituted chromans, processes for their preparation, their use as medicament or diagnostic aid, and medicament comprising them HOECHST AKTIENGESELLSCHAFT (DE) 2000-06-06 US disclosed
EP-0860440-A1 Sulfonamido substituted chromane derivatives with potassium channel blocking activity HOECHST AKTIENGESELLSCHAFT (DE) 1998-08-26 EP disclosed
EP-0807629-A1 Sulfonamido substituted chromane derivatives, method for their preparation, their use as medicaments or diagnostic agents aswell as medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-11-19 EP disclosed
EP-0188194-B1 AMINOACRYLIC ACID DERIVATIVES BAYER AG (DE) 1990-07-04 EP disclosed
US-4695646-A OXYQUINOLINECARBOXYLIC ACID INTERMEDIATES BAYER AKTIENGESELLSCHAFT (DE) 1987-09-22 US disclosed
EP-0188194-A2 Aminoacrylic acid derivatives BAYER AG (DE) 1986-07-23 EP disclosed
CN-86100221-A AMINOACRYLIC ACID DERIVATIVES 1986-07-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10611753-B2 Process for the manufacturing of medicaments ARSA, F8, CYP4A11 KCNQ3 1109/4885KCNQ2 1053/4885KCNE1 1776/4885
US-11066389-B2 Process for the manufacturing of medicaments ARSA, F8, CYP4A11 KCNQ3 1109/4885KCNQ2 1053/4885KCNE1 1776/4885
US-20200190061-A1 PROCESS FOR THE MANUFACTURING OF MEDICAMENTS ARSA, F8, CYP4A11 KCNQ3 1109/4885KCNQ2 1053/4885KCNE1 1776/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.