SCHEMBL6560425

SCHEMBL6560425

CCC1CCC2C(N)=Nc3cc(N(Cc4cccc(Cl)c4)C(=O)OC(C)(C)C)c(Cl)cc3C12

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 6/20 0.37
NOS1 P29475 6/20 0.37
NOS2 P35228 6/20 0.37
RIPK1 Q13546 1/20 0.34
GHSR Q92847 3/20 0.32
CPB2 Q96IY4 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
UCHL1 P09936 1/20 0.31
USP30 Q70CQ3 1/20 0.31
SLC6A9 P48067 2/20 0.31
KCNH2 Q12809 2/20 0.31
SLC6A5 Q9Y345 2/20 0.31
NPC1 O15118 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6069209 0.89 NOS3 (0.38) NOS3NOS1NOS2RIPK1GHSR
SCHEMBL6069550 0.80 NOS3 (0.39) NOS3NOS1NOS2RIPK1GHSR
SCHEMBL6069478 0.73 NOS3 (0.59) NOS3NOS1NOS2GHSR
SCHEMBL6069537 0.72 NOS3 (0.49) NOS3NOS1NOS2RIPK1GHSR
Hydrochloric Acid SCHEMBL6069850 0.72 NOS3 (0.52) NOS3NOS1NOS2
SCHEMBL6069538 0.72 NOS3 (0.57) NOS3NOS1NOS2GHSR
SCHEMBL6069204 0.70 NOS3 (0.56) NOS3NOS1NOS2GHSR
SCHEMBL6069521 0.70 NOS3 (0.50) NOS3NOS1NOS2RIPK1GHSR
SCHEMBL6069203 0.70 NOS3 (0.51) NOS3NOS1NOS2RIPK1GHSR
SCHEMBL6069425 0.69 NOS3 (0.46) NOS3NOS1NOS2SLC6A9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115708-B1 AMINOALKYL-3,4-DIHYDROQUINOLINE DERIVATES AS NO-SYNTHASE INHIBITORS SCHERING AG (DE) 2004-04-14 EP claimed