SCHEMBL6563177

SCHEMBL6563177

CS(=O)(=O)c1ccccc1N1N=C(C(F)(F)F)CC1c1ccc(F)c(F)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.55
PTGS1 P23219 11/20 0.55
PRKCZ Q05513 4/20 0.45
PDE5A O76074 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5693293 0.81 PTGS2 (0.73) PTGS2PTGS1PRKCZPDE5A
SCHEMBL5693452 0.79 PTGS2 (0.64) PTGS2PTGS1PRKCZPDE5A
SCHEMBL5693251 0.75 PTGS2 (0.64) PTGS2PTGS1PDE5A
SCHEMBL5693244 0.75 PTGS2 (0.64) PTGS2PTGS1PDE5A
SCHEMBL5856358 0.75 PTGS1 (0.73) PTGS2PTGS1
SCHEMBL5693286 0.74 PTGS2 (0.62) PTGS2PTGS1PDE5A
SCHEMBL5693262 0.73 PTGS2 (0.59) PTGS2PTGS1PRKCZPDE5A
SCHEMBL5693232 0.71 PTGS2 (0.76) PTGS2PTGS1PRKCZPDE5A
SCHEMBL5693239 0.70 PTGS2 (0.58) PTGS2PTGS1PDE5A
SCHEMBL5693347 0.70 PTGS2 (0.66) PTGS2PTGS1PRKCZPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1083171-B1 PYRAZOLINE DERIVATIVES, THEIR PREPARATION AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-04-28 EP claimed