SCHEMBL6563306

SCHEMBL6563306

COC(=O)[C@H](Cc1ccc(OCc2c(Cl)cccc2Cl)cc1)NC(=O)C1=C(C)/C(=C/C(=O)O)CCC1(C)C

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 18/20 0.47
ITGB1 P05556 4/20 0.47
PPARG P37231 1/20 0.43
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563309 1.00 ITGA4 (0.47) ITGA4ITGB1PPARGGAARAB9A
SCHEMBL6561247 0.94 ITGA4 (0.53) ITGA4ITGB1
SCHEMBL6561242 0.94 ITGA4 (0.53) ITGA4ITGB1
SCHEMBL6562500 0.90 ITGA4 (0.42) ITGA4ITGB1PPARG
SCHEMBL6562503 0.90 ITGA4 (0.42) ITGA4ITGB1PPARG
SCHEMBL6562539 0.85 ITGB1 (0.51) ITGA4ITGB1
SCHEMBL6562533 0.85 ITGB1 (0.51) ITGA4ITGB1
SCHEMBL6560288 0.78 ITGB1 (0.60) ITGA4ITGB1
SCHEMBL6560292 0.78 ITGB1 (0.60) ITGA4ITGB1
SCHEMBL6562552 0.75 ITGB1 (0.46) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144365-B1 INHIBITORS OF ALPHA-4 BETA-1 MEDIATED CELL ADHESION TANABE SEIYAKU CO (JP) 2004-03-17 EP disclosed