SCHEMBL6564643

SCHEMBL6564643

CCCS(=O)(=O)NCCCc1ccc(CNS(=O)(=O)CCC)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 3/20 0.39
HSD17B10 Q99714 3/20 0.39
TP53 P04637 1/20 0.39
ALDH1A1 P00352 3/20 0.38
HTT P42858 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6564987 0.92 SMN1; SMN2 (0.44) KDM4EHSD17B10TP53ALDH1A1HTT
SCHEMBL6562912 0.80 MEN1 (0.57) MEN1KMT2AKDM4EHSD17B10TP53
SCHEMBL6564635 0.78 GRIA4 (0.47) POLB
SCHEMBL6563391 0.77 MEN1 (0.54) MEN1KMT2AKDM4EHSD17B10TP53
SCHEMBL6563237 0.72 POLB (0.41) KMT2AALDH1A1SMN1; SMN2POLB
SCHEMBL6563319 0.71 SMN1; SMN2 (0.53) MEN1KMT2AKDM4EHSD17B10TP53
SCHEMBL5186035 0.71 MEN1 (0.50) MEN1KMT2AKDM4EHSD17B10TP53
SCHEMBL6565154 0.70 SMN1; SMN2 (0.50) MEN1KMT2AKDM4EHSD17B10TP53
SCHEMBL6562898 0.70 KMT2A (0.45) MEN1KMT2AKDM4EHSD17B10ALDH1A1
SCHEMBL29564150 0.70 CA9 (0.49) MEN1KMT2AHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296945-B1 SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2004-08-04 EP disclosed
US-6703425-B2 ADMINISTERING GLUTAMATE RECEPTOR POTENTIATOR TO TREAT PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY 2004-03-09 US disclosed
US-20030229102-A1 Sulfonamide derivatives ELI LILLY AND COMPANY 2003-12-11 US disclosed
EP-1296945-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2003-04-02 EP disclosed
WO-2001096289-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229102-A1 Sulfonamide derivatives GRIN1, GRIN2A, SLC1A2 MEN1 4129/4885KMT2A 723/4885KDM4E 2686/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.