SCHEMBL6563237

SCHEMBL6563237

CS(=O)(=O)NCCc1ccc(CNS(C)(=O)=O)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
NQO2 P16083 1/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.39
GRIA4 P48058 1/20 0.39
LMNA P02545 2/20 0.39
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 2/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
ADRA1A P35348 1/20 0.38
CA12 O43570 1/20 0.38
CA5A P35218 1/20 0.38
CA14 Q9ULX7 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14797697 0.83 TRPV1 (0.41) POLBTRPV1KMT2ALMNA
SCHEMBL14831186 0.82 ALDH1A1 (0.46) POLBTRPV1KMT2AALDH1A1LMNA
SCHEMBL6564982 0.81 GRIA4 (0.55) KMT2AALDH1A1GRIA4LMNACA1
SCHEMBL6564987 0.80 SMN1; SMN2 (0.44) ALDH1A1LMNACA1CA2CA9
SCHEMBL24632660 0.78 TRPV1 (0.44) TRPV1KMT2AALDH1A1LMNACA2
SCHEMBL13194426 0.76 ADRA2B (0.49) TRPV1KMT2ALMNAADRA2B
SCHEMBL13172655 0.76 P2RX7 (0.45) TRPV1LMNACA2
SCHEMBL21267602 0.74 TRPV1 (0.47) TRPV1GRIA4
SCHEMBL6564635 0.73 GRIA4 (0.47) POLBGRIA4LMNA
SCHEMBL14798069 0.73 FFAR1 (0.41) TRPV1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296945-B1 SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2004-08-04 EP disclosed
US-6703425-B2 ADMINISTERING GLUTAMATE RECEPTOR POTENTIATOR TO TREAT PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY 2004-03-09 US disclosed
US-20030229102-A1 Sulfonamide derivatives ELI LILLY AND COMPANY 2003-12-11 US disclosed
EP-1296945-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2003-04-02 EP disclosed
WO-2001096289-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229102-A1 Sulfonamide derivatives GRIN1, GRIN2A, SLC1A2 POLB 4443/4885TRPV1 300/4885NQO2 669/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.