SCHEMBL6565549

SCHEMBL6565549

O=C(Nc1ccccc1O)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 16/20 1.00
TSHR P16473 2/20 0.60
KDM4E B2RXH2 1/20 0.60
ALDH1A1 P00352 1/20 0.60
MAPT P10636 1/20 0.60
HPGD P15428 1/20 0.60
ALOX12 P18054 1/20 0.60
HTT P42858 1/20 0.60
ATM Q13315 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
HSD17B10 Q99714 1/20 0.60
RAB9A P51151 2/20 0.58
MAPK1 P28482 2/20 0.58
NPC1 O15118 1/20 0.56
GBA1 P04062 1/20 0.56
FAAH O00519 1/20 0.56
P2RX4 Q99571 1/20 0.56
P2RX7 Q99572 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6566257 0.83 EPHX2 (0.71) EPHX2TSHRKDM4EALDH1A1MAPT
SCHEMBL4357793 0.82 EPHX2 (0.70) EPHX2FAAH
SCHEMBL6567242 0.80 EPHX2 (0.67) EPHX2MAPTNPSR1
SCHEMBL4354504 0.80 EPHX2 (0.67) EPHX2MAPTNPSR1
SCHEMBL4350925 0.80 EPHX2 (0.67) EPHX2TSHRMAPTNPSR1RAB9A
SCHEMBL4341293 0.80 EPHX2 (0.67) EPHX2TSHRRAB9AMAPK1NPC1
SCHEMBL1420838 0.80 EPHX2 (1.00) EPHX2
SCHEMBL4000748 0.77 EPHX2 (0.62) EPHX2TSHRRAB9AMAPK1NPC1
SCHEMBL8064706 0.76 EPHX2 (0.61) EPHX2
SCHEMBL29450618 0.75 EPHX2 (0.66) EPHX2TSHRALDH1A1NPSR1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed