SCHEMBL6565667

SCHEMBL6565667

O=C(O)CNC(=O)c1nc2ccc(OCc3ccccc3)cc2cc1O

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 14/20 0.57
FTO Q9C0B1 5/20 0.51
EGLN3 Q9H6Z9 1/20 0.51
MEN1 O00255 1/20 0.49
HSP90AA1 P07900 1/20 0.49
KMT2A Q03164 1/20 0.49
KDM5B Q9UGL1 1/20 0.46
KDM2A Q9Y2K7 1/20 0.46
MAOB P27338 1/20 0.45
HIF1AN Q9NWT6 1/20 0.45
SPHK2 Q9NRA0 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
EGLN2 Q96KS0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6564152 0.91 EGLN1 (0.57) EGLN1FTOEGLN3KDM5BKDM2A
SCHEMBL6567196 0.90 EGLN1 (0.54) EGLN1FTOEGLN3MAOB
SCHEMBL1509109 0.85 EGLN1 (0.64) EGLN1FTO
SCHEMBL6566125 0.85 EGLN1 (0.52) EGLN1FTOEGLN3
SCHEMBL1509148 0.83 EGLN1 (0.50) EGLN1FTOEGLN3
SCHEMBL964980 0.83 EGLN1 (0.50) EGLN1FTOEGLN3
SCHEMBL6565865 0.82 EGLN1 (0.57) EGLN1FTOEGLN3HIF1AN
SCHEMBL8779216 0.82 EGLN1 (0.49) EGLN1FTOEGLN3
SCHEMBL8632085 0.82 HDAC8 (0.50) EGLN1MEN1HSP90AA1KMT2A
Hydrochloric Acid SCHEMBL6565656 0.81 EGLN1 (0.48) EGLN1FTOEGLN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765871-B1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors FIBROGEN INC (US) 2004-03-31 EP disclosed
US-5726305-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-10 US disclosed
US-5719164-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-17 US disclosed
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed
EP-0765871-A1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed