SCHEMBL6567196

SCHEMBL6567196

O=C(O)CNC(=O)c1nc2ccc(OCc3ccc(F)cc3)cc2cc1O

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 15/20 0.54
MAOB P27338 3/20 0.46
MAOA P21397 2/20 0.46
FTO Q9C0B1 2/20 0.46
EGLN3 Q9H6Z9 1/20 0.43
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565667 0.90 EGLN1 (0.57) EGLN1MAOBFTOEGLN3
SCHEMBL6566125 0.82 EGLN1 (0.52) EGLN1FTOEGLN3
SCHEMBL6564152 0.82 EGLN1 (0.57) EGLN1MAOBFTOEGLN3
SCHEMBL8779216 0.82 EGLN1 (0.49) EGLN1FTOEGLN3
Hydrochloric Acid SCHEMBL6565656 0.81 EGLN1 (0.48) EGLN1FTOEGLN3
SCHEMBL964980 0.81 EGLN1 (0.50) EGLN1FTOEGLN3
SCHEMBL1509148 0.81 EGLN1 (0.50) EGLN1FTOEGLN3
SCHEMBL8628981 0.80 EGLN1 (0.55) EGLN1FTO
SCHEMBL6567188 0.80 EGLN1 (0.47) EGLN1FTOEGLN3
SCHEMBL6565865 0.80 EGLN1 (0.57) EGLN1FTOEGLN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765871-B1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors FIBROGEN INC (US) 2004-03-31 EP disclosed
US-5726305-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-10 US disclosed
US-5719164-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-17 US disclosed
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed
EP-0765871-A1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
CN-1126203-A Substituted heterocyclic carboxamides, their preparation and their use as pharmaceuticals HOECHST AG (DE) 1996-07-10 CN disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed