SCHEMBL6567256

SCHEMBL6567256

CCCCOc1ccc2cc(O)c(C(=O)NCC(=O)O)nc2c1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 17/20 0.50
EGLN3 Q9H6Z9 3/20 0.49
FTO Q9C0B1 2/20 0.49
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
VEGFA P15692 2/20 0.46
FLT1 P17948 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL964980 0.91 EGLN1 (0.50) EGLN1EGLN3FTOALDH1A1LMNA
SCHEMBL6565270 0.88 EGLN1 (0.47) EGLN1EGLN3FTOALDH1A1LMNA
SCHEMBL6567272 0.88 EGLN1 (0.47) EGLN1EGLN3FTOALDH1A1LMNA
SCHEMBL6566238 0.88 EGLN1 (0.47) EGLN1EGLN3FTOALDH1A1LMNA
SCHEMBL1509148 0.86 EGLN1 (0.50) EGLN1EGLN3FTOVEGFAFLT1
SCHEMBL6564152 0.83 EGLN1 (0.57) EGLN1EGLN3FTO
SCHEMBL6565277 0.83 EGLN1 (0.47) EGLN1EGLN3FTOVEGFAFLT1
SCHEMBL8625366 0.81 EGLN1 (0.44) EGLN1EGLN3ALDH1A1LMNA
SCHEMBL6566125 0.81 EGLN1 (0.52) EGLN1EGLN3FTOVEGFAFLT1
SCHEMBL8633329 0.80 EGLN1 (0.54) EGLN1FTO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765871-B1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors FIBROGEN INC (US) 2004-03-31 EP disclosed
US-5726305-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-10 US disclosed
US-5719164-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-17 US disclosed
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed
EP-0765871-A1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
CN-1126203-A Substituted heterocyclic carboxamides, their preparation and their use as pharmaceuticals HOECHST AG (DE) 1996-07-10 CN disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed