SCHEMBL6568140

SCHEMBL6568140

CN(C)CC(=O)Nc1ccc(Sc2ccc(NC(=O)C(C)(O)C(F)(F)F)c(Cl)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 18/20 0.54
PDK2 Q15119 18/20 0.54
PDK3 Q15120 18/20 0.54
PDK4 Q16654 18/20 0.54
ABCB11 O95342 1/20 0.48
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6358481 1.00 PDK1 (0.54) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6570000 0.89 PDK1 (0.57) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6570004 0.89 PDK1 (0.57) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6570966 0.86 PDK1 (0.62) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6570960 0.86 PDK1 (0.62) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6571238 0.86 PDK1 (0.54) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6571231 0.86 PDK1 (0.54) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6569125 0.84 PDK1 (0.59) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6569113 0.84 PDK1 (0.59) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6571358 0.82 PDK1 (0.57) PDK1PDK2PDK3PDK4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082110-B1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2004-03-24 EP disclosed