SCHEMBL6569846

SCHEMBL6569846

CCOC(=O)c1cccc(-c2ccc(C(=O)Nc3ccc(OC)c(OCCN(C(C)C)C(C)C)c3)cc2)c1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 18/20 0.72
HTR2C P28335 1/20 0.71
CYP1A2 P05177 1/20 0.52
POLB P06746 1/20 0.52
CYP3A4 P08684 1/20 0.52
SLC2A1 P11166 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6570538 0.91 MCHR1 (0.74) MCHR1HTR2CCYP1A2POLBCYP3A4
Trifluoroacetic Acid SCHEMBL6570904 0.88 MCHR1 (0.71) MCHR1HTR2CCYP1A2POLBCYP3A4
SCHEMBL6927129 0.88 MCHR1 (0.93) MCHR1HTR2CCYP1A2POLBCYP3A4
SCHEMBL6926340 0.87 MCHR1 (0.92) MCHR1HTR2CSLC2A1
SCHEMBL6925891 0.87 MCHR1 (0.78) MCHR1HTR2CSLC2A1
SCHEMBL6927905 0.87 MCHR1 (0.78) MCHR1HTR2CCYP1A2POLBCYP3A4
SCHEMBL6924942 0.86 MCHR1 (0.75) MCHR1HTR2CSLC2A1
SCHEMBL6569788 0.85 MCHR1 (0.73) MCHR1HTR2CSLC2A1
Trifluoroacetic Acid SCHEMBL6569170 0.85 MCHR1 (0.72) MCHR1HTR2CSLC2A1
SCHEMBL6572159 0.85 MCHR1 (0.74) MCHR1HTR2CSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140072-B1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-04-14 EP claimed
EP-1140072-B1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-04-14 EP disclosed
WO-2004011427-A2 SUBSTITUTED BENZANILIDES AS MODULATORS OF THE CCR5 RECEPTOR SMITHKLINE BEECHAM CORPORATION (US) 2004-02-05 WO disclosed