SCHEMBL6569896

SCHEMBL6569896

C#Cc1cc(S(=O)(=O)c2ccc(S(C)(=O)=O)cc2)ccc1NC(=O)C(C)(O)C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 6/20 0.60
PDK2 Q15119 6/20 0.60
PDK3 Q15120 6/20 0.60
PDK4 Q16654 6/20 0.60
ABCC9 O60706 12/20 0.55
ABCC8 Q09428 12/20 0.55
KCNJ11 Q14654 12/20 0.55
KCNJ8 Q15842 12/20 0.55
ABCB11 O95342 1/20 0.53
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6569892 1.00 PDK1 (0.60) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL6345815 0.85 PDK1 (0.55) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL6345819 0.85 PDK1 (0.55) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL6569996 0.84 PDK1 (0.65) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL6570002 0.84 PDK1 (0.65) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL6569823 0.83 PDK1 (0.86) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6358430 0.83 PDK1 (0.63) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL6358427 0.83 PDK1 (0.63) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL6569819 0.83 PDK1 (0.86) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6351331 0.80 PDK1 (0.60) PDK1PDK2PDK3PDK4ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082110-B1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2004-03-24 EP disclosed