SCHEMBL6571265

SCHEMBL6571265

COc1ccc(C(=O)Nc2ccc(NC(=O)C(C)(O)C(F)(F)F)c(Cl)c2)cc1

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 19/20 0.68
PDK2 Q15119 19/20 0.68
PDK3 Q15120 19/20 0.68
PDK4 Q16654 19/20 0.68
NPC1 O15118 1/20 0.51
TP53 P04637 1/20 0.51
ALOX15 P16050 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571257 1.00 PDK1 (0.68) PDK1PDK2PDK3PDK4NPC1
SCHEMBL3787237 0.85 MAPT (0.68) NPC1TP53ALOX15RAB9ASMN1; SMN2
SCHEMBL5736882 0.83 PDK1 (0.62) PDK1PDK2PDK3PDK4
SCHEMBL6571391 0.82 PDK1 (0.61) PDK1PDK2PDK3PDK4
SCHEMBL5749870 0.80 PDK1 (0.64) PDK1PDK2PDK3PDK4
SCHEMBL4624630 0.80 PDK1 (0.61) PDK1PDK2PDK3PDK4
SCHEMBL4624625 0.80 PDK1 (0.61) PDK1PDK2PDK3PDK4
SCHEMBL6568163 0.80 PDK1 (0.71) PDK1PDK2PDK3PDK4
SCHEMBL6568929 0.80 PDK1 (0.71) PDK1PDK2PDK3PDK4
SCHEMBL6568923 0.80 PDK1 (0.71) PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082110-B1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2004-03-24 EP disclosed