SCHEMBL6571612

SCHEMBL6571612

CC(O)(C(=O)Nc1ccc(S(=O)(=O)c2ccc(F)c(Cl)c2)cc1Cl)C(F)(F)F

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 18/20 0.74
PDK2 Q15119 18/20 0.74
PDK3 Q15120 18/20 0.74
PDK4 Q16654 18/20 0.74
ABCB11 O95342 1/20 0.70
PTGES2 Q9H7Z7 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571603 1.00 PDK1 (0.74) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6571262 0.94 PDK1 (0.72) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6571268 0.94 PDK1 (0.72) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL4609233 0.91 PDK1 (0.74) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL4609236 0.91 PDK1 (0.74) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6568935 0.89 PDK1 (0.75) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6568943 0.89 PDK1 (0.75) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6571208 0.88 PDK1 (0.74) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL6571201 0.88 PDK1 (0.74) PDK1PDK2PDK3PDK4ABCB11
SCHEMBL4609853 0.88 PDK1 (0.74) PDK1PDK2PDK3PDK4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082110-B1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2004-03-24 EP disclosed