SCHEMBL6571664

SCHEMBL6571664

NCCNCn1cc(Cl)c(=O)[nH]c1=O

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.48
GRIA2 P42262 1/20 0.48
GRIA4 P48058 1/20 0.48
GRIK5 Q16478 1/20 0.48
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571691 0.81 GRIA1 (0.48) GRIA1GRIA2GRIA4GRIK5
SCHEMBL6571672 0.81 KMT2A (0.48) GRIA1GRIA2GRIA4GRIK5HPGD
SCHEMBL6572744 0.77 GRIA1 (0.49) GRIA1GRIA2GRIA4GRIK5HPGD
SCHEMBL11254252 0.71 GRIA1 (0.53) GRIA1GRIA2GRIA4GRIK5HPGD
SCHEMBL2353226 0.69 GRIA1 (0.48) GRIA1GRIA2GRIA4GRIK5
SCHEMBL19711624 0.68 GRIA1 (0.54) GRIA1GRIA2GRIA4GRIK5HPGD
SCHEMBL5116514 0.68 GRIA1 (0.54) GRIA1GRIA2GRIA4GRIK5
SCHEMBL14208548 0.67 DTYMK (0.56)
SCHEMBL30423828 0.67 GRIA1 (0.60) GRIA1GRIA2GRIA4GRIK5
SCHEMBL6570527 0.66 GRIA1 (0.48) GRIA1GRIA2GRIA4GRIK5HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0884051-B1 CANCEROUS METASTASIS INHIBITORS CONTAINING URACIL DERIVATIVES TAIHO PHARMACEUTICAL CO LTD (JP) 2004-12-15 EP disclosed
EP-0763529-B1 URACIL DERIVATIVES, AND ANTITUMOR EFFECT POTENTIATOR AND ANTITUMOR AGENT CONTAINING THE SAME TAIHO PHARMACEUTICAL CO LTD (JP) 2003-07-23 EP disclosed
US-6294535-B1 TREATING CANCER, WHICH COMPRISES ADMINISTERING TO A PATIENT IN NEED OF TREATMENT AN EFFECTIVE AMOUNT OF A URACIL DERIVATIVE TAIHO PHARMACEUTICAL CO., LTD. (JP) 2001-09-25 US disclosed
US-6255314-B1 Cancerous metastasis inhibitors containing uracil derivatives TAIHO CHARMACEUTICAL CO., LTD. (JP) 2001-07-03 US disclosed
US-6159969-A Uracil derivatives, and antitumor effect potentiator and antitumor agent containing the same TAIHO PHARMACEUTICAL CO., LTD. (JP) 2000-12-12 US disclosed
EP-0884051-A1 CANCEROUS METASTASIS INHIBITORS CONTAINING URACIL DERIVATIVES TAIHO PHARMACEUTICAL COMPANY LIMITED (JP) 1998-12-16 EP disclosed
US-5744475-A 4-N-HET-METHYLURACIL DERIVATIVES; THYMIDINE PHOSPHORYLASE INHIBITORS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1998-04-28 US disclosed
EP-0763529-A1 URACIL DERIVATIVES, AND ANTITUMOR EFFECT POTENTIATOR AND ANTITUMOR AGENT CONTAINING THE SAME TAIHO PHARMACEUTICAL COMPANY LIMITED (JP) 1997-03-19 EP disclosed