SCHEMBL6571859

SCHEMBL6571859

Nc1cccc(-c2cc(N)ccc2NCC(O)CO)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
MAOA P21397 1/20 0.36
MAP4K4 O95819 1/20 0.36
CHEK1 O14757 1/20 0.35
CDK1 P06493 1/20 0.35
IRAK1 P51617 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
IDH2 P48735 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571461 0.93 CHEK1 (0.41) MAOACHEK1CDK1PTGDR2
SCHEMBL6572232 0.92 PIK3CG (0.38) ALDH1A1MAP4K4CHEK1CDK1IRAK1
Hydrochloric Acid SCHEMBL6572537 0.91 CHEK1 (0.40) MAOACHEK1CDK1PTGDR2
SCHEMBL6571398 0.91 TAAR1 (0.41) IDH2
SCHEMBL6571424 0.91 EGFR (0.39) KDM4EMAPTCHEK1CDK1IRAK1
SCHEMBL6572450 0.91 ADORA1 (0.37) ALDH1A1
SCHEMBL6574847 0.90 PDE3B (0.37) CHEK1CDK1
SCHEMBL6572042 0.88 PDE3B (0.34) CHEK1CDK1IDH2
SCHEMBL6570761 0.88 DYRK3 (0.35) CHEK1CDK1IRAK1IRAK4PTGDR2
SCHEMBL6570890 0.88 IDH2 (0.48) ALDH1A1IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed