SCHEMBL6572042

SCHEMBL6572042

Nc1cc(N)cc(-c2cc(N)ccc2NCC(O)CO)c1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
AR P10275 2/20 0.33
VDR P11473 2/20 0.33
CHEK1 O14757 1/20 0.32
CDK1 P06493 1/20 0.32
CYP1A2 P05177 1/20 0.30
IDH2 P48735 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6574847 0.92 PDE3B (0.37) PDE3BPDE3AARVDRCHEK1
SCHEMBL6574582 0.92 PDE3B (0.32) PDE3BPDE3AARVDR
SCHEMBL6572447 0.90 ADRB2 (0.33) PDE3BPDE3AARVDR
SCHEMBL6571461 0.90 CHEK1 (0.41) CHEK1CDK1
SCHEMBL6571859 0.88 KDM4E (0.37) CHEK1CDK1IDH2
Hydrochloric Acid SCHEMBL6572537 0.88 CHEK1 (0.40) CHEK1CDK1
SCHEMBL6573407 0.88 USP7 (0.36) PDE3BPDE3AARVDR
SCHEMBL6571878 0.87 CYP1A2 (0.38) PDE3BPDE3ACYP1A2
SCHEMBL6571824 0.87 CYP1A2 (0.34) PDE3BPDE3AARVDRCYP1A2
SCHEMBL6571431 0.87 AR (0.36) PDE3BPDE3AARVDRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed