SCHEMBL6572098

SCHEMBL6572098

COc1ccc(CCN(C)CCOc2ccc([N+](=O)[O-])cc2OCc2ccccc2)cc1OC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.62
CYP3A4 P08684 3/20 0.62
CYP2D6 P10635 3/20 0.62
BLM P54132 2/20 0.62
CYP2C9 P11712 2/20 0.62
KDM4E B2RXH2 1/20 0.62
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
KCNH2 Q12809 3/20 0.50
ALDH1A1 P00352 2/20 0.49
CYP19A1 P11511 2/20 0.49
PMP22 Q01453 1/20 0.49
MAPT P10636 2/20 0.48
HTR1A P08908 2/20 0.48
ADRA1D P25100 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575943 0.84 CYP1A2 (0.56) CYP1A2CYP3A4CYP2D6BLMCYP2C9
SCHEMBL6573041 0.83 CYP1A2 (0.55) CYP1A2CYP3A4CYP2D6BLMCYP2C9
SCHEMBL6571843 0.83 CYP1A2 (0.55) CYP1A2CYP3A4CYP2D6BLMCYP2C9
Hydrochloric Acid SCHEMBL6571816 0.83 BLM (0.57) CYP1A2CYP3A4CYP2D6BLMCYP2C9
SCHEMBL6574454 0.83 MAPT (0.60) CYP1A2CYP3A4CYP2D6BLMCYP2C9
Hydrochloric Acid SCHEMBL6573751 0.82 BLM (0.56) CYP1A2CYP3A4CYP2D6BLMCYP2C9
SCHEMBL5929724 0.82 MAPT (0.67) CYP1A2CYP3A4CYP2D6CYP2C9KDM4E
SCHEMBL30721937 0.82 MAPT (0.67) CYP1A2CYP3A4CYP2D6CYP2C9MEN1
SCHEMBL30354869 0.82 MAPT (0.67) CYP1A2CYP3A4CYP2D6CYP2C9KDM4E
SCHEMBL2063456 0.82 MAPT (0.67) CYP1A2CYP3A4CYP2D6CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775689-B9 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RES LABS (KR) 2004-09-15 EP disclosed
EP-0775689-B1 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RES LABS (KR) 2003-09-03 EP disclosed
US-6057358-A POTASSIUM CHANNEL BLOCKING ANTIARRHYTHMIC DRUGS WITH LESS SIDE EFFECTS C&C RESEARCH LABS. (KR) 2000-05-02 US disclosed
EP-0775689-A1 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RESEARCH LABS. (KR) 1997-05-28 EP disclosed