SCHEMBL6571843

SCHEMBL6571843

COc1ccc(CCN(C)CCOc2ccc([N+](=O)[O-])cc2N(C)C)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 2/20 0.55
CDC25C P30307 2/20 0.55
KCNH2 Q12809 4/20 0.55
BLM P54132 2/20 0.54
PMP22 Q01453 1/20 0.54
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
THRB P10828 1/20 0.48
APEX1 P27695 1/20 0.48
RECQL P46063 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
MAPT P10636 3/20 0.47
AOC3 Q16853 1/20 0.44
NPC1 O15118 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575943 0.88 CYP1A2 (0.56) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
SCHEMBL6574454 0.87 MAPT (0.60) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
SCHEMBL6573041 0.87 CYP1A2 (0.55) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
Hydrochloric Acid SCHEMBL6571816 0.87 BLM (0.57) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
Hydrochloric Acid SCHEMBL6573751 0.86 BLM (0.56) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
SCHEMBL6573083 0.86 KCNH2 (0.76) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
Hydrochloric Acid SCHEMBL6574014 0.84 PMP22 (0.53) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
SCHEMBL6574500 0.83 KCNH2 (0.50) CYP1A2CYP3A4CYP2D6CDC25CKCNH2
SCHEMBL6572098 0.83 CYP1A2 (0.62) CYP1A2CYP3A4CYP2D6KCNH2BLM
SCHEMBL6572877 0.82 KCNH2 (0.54) CYP1A2CYP3A4CYP2D6CDC25CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775689-B9 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RES LABS (KR) 2004-09-15 EP disclosed
EP-0775689-B1 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RES LABS (KR) 2003-09-03 EP disclosed
US-6057358-A POTASSIUM CHANNEL BLOCKING ANTIARRHYTHMIC DRUGS WITH LESS SIDE EFFECTS C&C RESEARCH LABS. (KR) 2000-05-02 US disclosed
EP-0775689-A1 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RESEARCH LABS. (KR) 1997-05-28 EP disclosed