SCHEMBL6573776

SCHEMBL6573776

COC(=O)[C@H](Cc1ccc(-n2cccn2)cc1)NC(=O)[C@@H](CSC(C)=O)C(C)C

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FCER2 P06734 1/20 0.42
ALDH1A1 P00352 1/20 0.41
THRB P10828 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TSHR P16473 1/20 0.40
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
CAPN1 P07384 1/20 0.36
TP53 P04637 1/20 0.36
MDM4 O15151 1/20 0.36
MDM2 Q00987 1/20 0.36
POLB P06746 1/20 0.36
GFER P55789 1/20 0.36
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572061 0.82 KDM4E (0.44) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL6572892 0.77 MME (0.54)
SCHEMBL7262826 0.77 MME (0.54)
SCHEMBL7262844 0.75 KLK5 (0.50)
SCHEMBL7262965 0.75 MAPT (0.36) MAPTTP53POLB
SCHEMBL6575357 0.74 MAPT (0.44) ALDH1A1KDM4EMAPTTP53
SCHEMBL6575361 0.74 MAPT (0.44) ALDH1A1KDM4EMAPTTP53
Hydrochloric Acid SCHEMBL6574263 0.73 MAPT (0.43) ALDH1A1KDM4EMAPTTP53
SCHEMBL16632664 0.69 MAPT (0.42) ALDH1A1KDM4EMAPTTP53
SCHEMBL8165462 0.69 CYP2C9 (0.61) ALDH1A1THRBCYP2C9CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474405-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2004-11-10 EP disclosed
WO-2003104200-A1 N-MERCAPTOACYL PHENYALANINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 2003-12-18 WO disclosed
WO-2003068725-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-08-21 WO disclosed