SCHEMBL6572061

SCHEMBL6572061

COC(=O)[C@H](Cc1ccc(-n2cccn2)cc1)NC(C)=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
ATM Q13315 2/20 0.43
POLB P06746 2/20 0.43
CTSD P07339 2/20 0.43
BACE1 P56817 2/20 0.43
GFER P55789 1/20 0.43
TACR1 P25103 1/20 0.43
CAPN1 P07384 1/20 0.43
ALDH1A1 P00352 1/20 0.43
THRB P10828 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262844 0.85 KLK5 (0.50)
SCHEMBL6575361 0.84 MAPT (0.44) KDM4EALDH1A1PIK3CDPIK3CAPIK3CB
SCHEMBL6575357 0.84 MAPT (0.44) KDM4EALDH1A1PIK3CDPIK3CAPIK3CB
Hydrochloric Acid SCHEMBL6574263 0.83 MAPT (0.43) KDM4EALDH1A1PIK3CDPIK3CAPIK3CB
SCHEMBL6573776 0.82 FCER2 (0.42) KDM4EATMPOLBGFERCAPN1
SCHEMBL16632664 0.79 MAPT (0.42) KDM4EALDH1A1MAPT
SCHEMBL7256083 0.78 CAPN1 (0.46) KDM4ECAPN1ALDH1A1PIK3CDPIK3CA
Hydrochloric Acid SCHEMBL6574264 0.77 CAPN1 (0.45) KDM4ECAPN1ALDH1A1PIK3CDPIK3CA
SCHEMBL18472617 0.76 NOS2 (0.65) KDM4EATMTACR1ALDH1A1THRB
SCHEMBL7221067 0.76 NOS2 (0.65) KDM4EATMTACR1ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474405-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2004-11-10 EP disclosed
WO-2003068725-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-08-21 WO disclosed