SCHEMBL6575289

SCHEMBL6575289

Cc1noc([C@H]2O[C@@H](n3cnc4c(N[C@@H]5CCC[C@H]5O)ncnc43)[C@H](O)[C@@H]2O)n1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 11/20 0.64
ADORA1 P30542 8/20 0.64
ADORA3 P0DMS8 6/20 0.64
ADORA2B P29275 4/20 0.64
CYP2D6 P10635 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6574959 0.89 ADORA3 (0.62) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6574645 0.88 ADORA1 (0.51) ADORA2AADORA1ADORA3ADORA2BCYP2D6
SCHEMBL6572906 0.88 ADORA3 (0.60) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6573829 0.86 ADORA1 (0.66) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6797276 0.85 ADORA2A (0.65) ADORA2AADORA1ADORA3ADORA2BCYP2D6
SCHEMBL6572451 0.85 ADORA2A (0.62) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6574622 0.85 ADORA2A (0.65) ADORA2AADORA1ADORA3ADORA2BCYP2D6
SCHEMBL6574214 0.84 ADORA2A (0.57) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6573819 0.82 ADORA3 (0.63) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6576651 0.82 ADORA1 (0.65) ADORA2AADORA1ADORA3ADORA2BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090019-B1 ADENOSINE DERIVATIVES GLAXO GROUP LTD (GB) 2004-09-29 EP disclosed
EP-1447407-A1 Adenosine derivatives GLAXO GROUP LIMITED (GB) 2004-08-18 EP disclosed