SCHEMBL6575763

SCHEMBL6575763

BrCCOc1ccc(-c2ncc[nH]2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.71
CYP2D6 P10635 4/20 0.71
CYP1A2 P05177 3/20 0.71
CYP19A1 P11511 2/20 0.71
CYP2C9 P11712 2/20 0.71
CYP2C19 P33261 2/20 0.71
KCNH2 Q12809 1/20 0.58
HRH3 Q9Y5N1 1/20 0.58
NISCH Q9Y2I1 2/20 0.51
MTOR P42345 1/20 0.50
ADK P55263 1/20 0.50
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
ACHE P22303 2/20 0.39
HPGD P15428 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALOX12 P18054 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723343 0.83 CYP1A2 (0.88) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL4723390 0.83 CYP2D6 (1.00) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL14599590 0.82 CYP1A2 (0.70) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL6941842 0.81 CYP1A2 (0.73) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL12462292 0.81 CYP1A2 (0.72) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL6002465 0.80 CYP2D6 (0.91) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL3407136 0.79 CYP1A2 (0.76) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL722191 0.78 NISCH (0.78) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL15764580 0.75 CYP1A2 (0.65) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
Methyl Alcohol SCHEMBL10336733 0.75 CYP1A2 (0.69) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775689-B9 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RES LABS (KR) 2004-09-15 EP disclosed
EP-0775689-B1 NOVEL AMINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF AS ANTIARRHYTHMIC C & C RES LABS (KR) 2003-09-03 EP disclosed