SCHEMBL6576406

SCHEMBL6576406

Cn1cc(NC(=O)c2nc(NC(=O)c3nc(NC(=O)c4nccn4C)cn3C)cn2C)cc1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.46
ERBB2 P04626 1/20 0.42
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
GRM1 Q13255 4/20 0.40
GRM4 Q14833 6/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
KDM4E B2RXH2 2/20 0.38
POLB P06746 2/20 0.38
NTRK1 P04629 1/20 0.38
MAPT P10636 1/20 0.37
NR3C1 P04150 3/20 0.36
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25252633 0.98 NAMPT (0.45) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL5331486 0.92 NAMPT (0.46) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL30125632 0.92 NAMPT (0.46) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL2072460 0.91 NAMPT (0.54) NAMPTGRM1GRM4ROCK2ROCK1
SCHEMBL14388685 0.90 NAMPT (0.46) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL6433630 0.89 NAMPT (0.45) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL31615222 0.88 HDAC1 (0.51) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL23728665 0.88 HDAC1 (0.57) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL23728539 0.88 HDAC1 (0.57) NAMPTERBB2HDAC1HDAC2HDAC8
SCHEMBL20485621 0.88 NAMPT (0.52) NAMPTGRM1GRM4ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430028-A2 AROMATIC AND HETEROAROMATIC ACID HALIDES FOR SYNTHESIZING POLYAMIDES Pharmacia Corporation (US) 2004-06-23 EP disclosed
EP-1421056-A1 (ALPHA)-HALOENAMINE REAGENTS Pharmacia Corporation (US) 2004-05-26 EP disclosed
WO-2003020684-A1 (ALPHA)-HALOENAMINE REAGENTS PHARMACIA CORPORATION (US) 2003-03-13 WO disclosed
WO-2003018552-A2 AROMATIC AND HETEROAROMATIC ACID HALIDES FOR SYNTHESIZING POLYAMIDES PHARMACIA CORPORATION (US) 2003-03-06 WO disclosed