SCHEMBL6578742

SCHEMBL6578742

[CH2]c1cccc(-c2n[nH]c(-c3ccc(OC)cc3)n2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.67
NR1H3 Q13133 5/20 0.67
ADORA2A P29274 3/20 0.58
ADORA1 P30542 3/20 0.58
KDM4E B2RXH2 1/20 0.51
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MAPT P10636 2/20 0.49
KMT2A Q03164 2/20 0.49
ATAD2 Q6PL18 1/20 0.49
MEN1 O00255 1/20 0.49
TSHR P16473 1/20 0.49
HTT P42858 1/20 0.49
DCUN1D1 Q96GG9 1/20 0.46
TP53 P04637 1/20 0.45
DGAT1 O75907 2/20 0.44
LMNA P02545 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17279684 0.84 NR1H2 (0.67) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6579126 0.83 NR1H2 (0.49) NR1H2NR1H3ADORA2AADORA1NPC1
SCHEMBL15025693 0.83 NR1H2 (0.73) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL15117068 0.82 KDM4E (0.67) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6581499 0.81 NR1H2 (0.50) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6581439 0.81 NR1H2 (0.52) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6578706 0.81 NR1H2 (0.62) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6581717 0.81 NR1H2 (0.62) NR1H2NR1H3ADORA2AADORA1KDM4E
Hydrochloric Acid SCHEMBL6580735 0.80 NR1H2 (0.61) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6582914 0.79 NR1H2 (0.60) NR1H2NR1H3ADORA2AADORA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed