SCHEMBL6581499

SCHEMBL6581499

[CH2]c1cccc(-c2n[nH]c(-c3ccc(OC)c(F)c3)n2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.50
NR1H3 Q13133 4/20 0.50
ADORA2A P29274 3/20 0.50
ADORA1 P30542 2/20 0.50
KDM4E B2RXH2 1/20 0.46
HSD17B10 Q99714 1/20 0.46
LCK P06239 2/20 0.45
BTK Q06187 2/20 0.45
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
MEN1 O00255 2/20 0.41
NPC1 O15118 2/20 0.41
ALDH1A1 P00352 2/20 0.41
RAB9A P51151 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582892 0.86 ADORA2A (0.41) NR1H2NR1H3ADORA2AADORA1LCK
SCHEMBL6578586 0.86 S1PR1 (0.44) NR1H2NR1H3ADORA2AADORA1LCK
SCHEMBL6581439 0.85 NR1H2 (0.52) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6578742 0.81 NR1H2 (0.67) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6580942 0.81 HTR7 (0.46) NR1H2NR1H3ADORA2AADORA1KDM4E
Hydrochloric Acid SCHEMBL6581027 0.80 HTR7 (0.46) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL28095606 0.80 KDM4E (0.55) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6580708 0.79 ADORA2A (0.44) NR1H2NR1H3ADORA2AADORA1KDM4E
SCHEMBL6578503 0.78 ADORA2A (0.62) NR1H2NR1H3ADORA2AADORA1LCK
Hydrochloric Acid SCHEMBL6582961 0.77 ADORA2A (0.61) NR1H2NR1H3ADORA2AADORA1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed