SCHEMBL6578760

SCHEMBL6578760

CCn1nc(-c2ccc(OC)cc2)nc1-c1cccc(CN2CCCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 6/20 0.51
NR1H3 Q13133 3/20 0.50
NR1H2 P55055 2/20 0.50
DRD2 P14416 1/20 0.50
DRD4 P21917 1/20 0.50
DRD3 P35462 1/20 0.50
ACP1 P24666 3/20 0.46
TGM2 P21980 1/20 0.45
TGM1 P22735 1/20 0.45
CASP3 P42574 1/20 0.45
TGM3 Q08188 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
S1PR1 P21453 1/20 0.45
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6581009 0.99 AVPR1B (0.50) AVPR1BNR1H3NR1H2DRD2DRD4
Hydrochloric Acid SCHEMBL6580578 0.95 NR1H3 (0.54) AVPR1BNR1H3NR1H2DRD2DRD4
Hydrochloric Acid SCHEMBL6578233 0.90 NR1H3 (0.62) AVPR1BNR1H3NR1H2DRD2DRD4
SCHEMBL6578508 0.87 ADORA2A (0.55) AVPR1BDRD2DRD4DRD3ACP1
Hydrochloric Acid SCHEMBL6580767 0.87 AVPR1B (0.56) AVPR1BNR1H3NR1H2DRD2DRD4
Hydrochloric Acid SCHEMBL6581333 0.87 AVPR1B (0.47) AVPR1BNR1H3NR1H2DRD2DRD4
Hydrochloric Acid SCHEMBL6578595 0.86 ADORA2A (0.54) AVPR1BDRD2DRD4DRD3ACP1
Hydrochloric Acid SCHEMBL6584023 0.86 NR1H3 (0.68) AVPR1BNR1H3NR1H2DRD2DRD4
SCHEMBL17280134 0.84 NR1H3 (0.57) AVPR1BNR1H3NR1H2TGM2TGM1
Hydrochloric Acid SCHEMBL6581135 0.83 NR1H2 (0.56) AVPR1BNR1H3NR1H2DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US claimed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP claimed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed