SCHEMBL6579500

SCHEMBL6579500

CCCCCCCCOc1c(O)c2ccc(N)cc2n(C)c1=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TTR P02766 2/20 0.47
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 2/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
GSK3B P49841 9/20 0.44
TSHR P16473 1/20 0.40
MAPT P10636 3/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TYMS P04818 1/20 0.39
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR2 P34972 1/20 0.38
GPR84 Q9NQS5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8004161 1.00 TTR (0.47) TTRALDH1A1KDM4EHPGDHSD17B10
SCHEMBL6581772 0.95 TTR (0.49) TTRALDH1A1KDM4EHPGDHSD17B10
SCHEMBL7999367 0.91 TTR (0.47) TTRALDH1A1KDM4EHPGDHSD17B10
SCHEMBL7974971 0.91 ALDH1A1 (0.45) TTRALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8001545 0.89 TSHR (0.43) TTRALDH1A1KDM4EHPGDHSD17B10
SCHEMBL7988809 0.89 TSHR (0.43) TTRALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8001735 0.88 KDM4E (0.44) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL7997334 0.88 KDM4E (0.46) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL7999961 0.88 KDM4E (0.46) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL7998893 0.88 KDM4E (0.46) ALDH1A1KDM4EHPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1158265-C Quinoline ketone derivant and antianaphylaction using same as active substance ���ձ���ī��ѧ��ҵ��ʽ���� 2004-07-21 CN disclosed
EP-0927718-B1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK & CHEMICALS (JP) 2004-02-25 EP disclosed
CN-1095834-C Quinolinone derivatives and antiallergic agent containing said quinolinone derivatives as active ingredient DAINIPPON INK & CHEMICALS (JP) 2002-12-11 CN disclosed
US-6271416-B1 O-(HYDROCARBONOXYACETAMIDO)BENZOIC ACID DERIVATIVES AS INTERMEDIATES DAINIPPON INK AND CHEMICALS, INC. (JP) 2001-08-07 US disclosed
CN-1275564-A Quinoline ketone derivant and antianaphylaction using same as active substance DAINIPPON INK & CHEMICALS (JP) 2000-12-06 CN disclosed
US-6136822-A ETHER, HYDROXY QUINOLINONE COMPOUNDS DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-10-24 US disclosed
US-6114352-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-09-05 US disclosed
EP-0785190-B1 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK & CHEMICALS (JP) 2000-08-16 EP disclosed
US-5942521-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-08-24 US disclosed
EP-0927718-A1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-07-07 EP disclosed
CN-1163268-A Quinolinone derivatives and antiallergic agent containing said quinolinone derivatives as active ingredient LAINIPPON INK AND CHEMICALC IN (JP) 1997-10-29 CN disclosed
EP-0785190-A2 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1997-07-23 EP disclosed