SCHEMBL6580651

SCHEMBL6580651

CNC1CN(c2c(F)cc3c(=O)c(C(=O)O)cn(-c4cc(N)c(F)cc4F)c3c2C)C1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.49
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
TOP2A P11388 11/20 0.45
TOP1 P11387 8/20 0.45
TOP2B Q02880 5/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578732 0.94 KCNH2 (0.48) KCNH2CYP3A4CYP2C9TOP2ATOP1
SCHEMBL21341272 0.91 KCNH2 (0.47) KCNH2CYP3A4CYP2C9TOP2ATOP1
SCHEMBL7007374 0.90 CYP3A4 (0.58) CYP3A4CYP2C9TOP2ATOP1TOP2B
SCHEMBL6580734 0.90 CYP3A4 (0.56) KCNH2CYP3A4CYP2C9TOP2ATOP1
SCHEMBL6578454 0.90 KCNH2 (0.48) KCNH2CYP3A4CYP2C9TOP2ATOP1
SCHEMBL6581505 0.84 KCNH2 (0.51) KCNH2CYP3A4CYP2C9TOP2ATOP1
SCHEMBL6578831 0.84 CYP3A4 (0.54) KCNH2CYP3A4CYP2C9TOP2ATOP1
SCHEMBL6578566 0.84 KCNH2 (0.47) KCNH2CYP3A4CYP2C9TOP2ATOP1
SCHEMBL20912595 0.83 TOP2A (0.43) CYP3A4CYP2C9TOP2ATOP1TOP2B
SCHEMBL20912556 0.82 KCNH2 (0.46) KCNH2CYP3A4CYP2C9TOP2ATOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0897919-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND ANTIBACTERIAL AGENTS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2004-06-16 EP disclosed
US-6211375-B1 IMPROVED INTESTINAL ABSORPTION WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0897919-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND ANTIBACTERIAL AGENTS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-02-24 EP disclosed