SCHEMBL6582816

SCHEMBL6582816

COc1ccc(-c2nc(-c3cccc(CNC(C)=O)c3)n[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.54
NR1H3 Q13133 1/20 0.54
AURKA O14965 1/20 0.52
AURKB Q96GD4 1/20 0.52
LMNA P02545 4/20 0.51
TP53 P04637 4/20 0.51
CPT2 P23786 1/20 0.49
CPT1A P50416 1/20 0.49
HPGD P15428 1/20 0.48
ADORA2A P29274 2/20 0.48
ADORA1 P30542 1/20 0.48
MAPT P10636 3/20 0.48
ADORA3 P0DMS8 1/20 0.47
DGAT1 O75907 1/20 0.46
ROCK2 O75116 1/20 0.46
CHRM3 P20309 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580756 0.85 NR1H2 (0.60) NR1H2NR1H3LMNATP53HPGD
Hydrochloric Acid SCHEMBL6581037 0.84 NR1H2 (0.58) NR1H2NR1H3LMNATP53HPGD
Hydrochloric Acid SCHEMBL6584260 0.82 NR1H2 (0.53) NR1H2NR1H3LMNATP53HPGD
SCHEMBL6578706 0.81 NR1H2 (0.62) NR1H2NR1H3LMNATP53HPGD
Hydrochloric Acid SCHEMBL6580735 0.80 NR1H2 (0.61) NR1H2NR1H3LMNATP53HPGD
Hydrochloric Acid SCHEMBL6584025 0.79 NR1H2 (0.52) NR1H2NR1H3LMNATP53HPGD
SCHEMBL6580995 0.79 ALDH1A1 (0.52) NR1H2NR1H3LMNAADORA2AADORA1
SCHEMBL6582914 0.79 NR1H2 (0.60) NR1H2NR1H3LMNAHPGDADORA2A
Hydrochloric Acid SCHEMBL6580524 0.78 NR1H2 (0.58) NR1H2NR1H3HPGDADORA2AADORA1
SCHEMBL6578180 0.77 DRD4 (0.51) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed