SCHEMBL6583066

SCHEMBL6583066

COc1ccc(-c2nc(-c3cccc(CN(C)C)c3)n(C(F)F)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 2/20 0.43
AVPR1B P47901 3/20 0.42
HTR7 P34969 1/20 0.41
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
TNK2 Q07912 1/20 0.41
HSD17B2 P37059 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA1 P30542 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
TP53 P04637 2/20 0.37
S1PR1 P21453 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
EGFR P00533 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6582405 0.89 AVPR1B (0.44) ACP1AVPR1BHTR7NR1H2NR1H3
Hydrochloric Acid SCHEMBL6580886 0.85 NR1H2 (0.46) ACP1AVPR1BHTR7NR1H2NR1H3
Hydrochloric Acid SCHEMBL6580906 0.85 NR1H2 (0.46) ACP1AVPR1BHTR7NR1H2NR1H3
SCHEMBL6584053 0.84 ACP1 (0.46) ACP1AVPR1BHTR7NR1H2NR1H3
Hydrochloric Acid SCHEMBL6580533 0.84 ACP1 (0.45) ACP1AVPR1BHTR7NR1H2NR1H3
SCHEMBL6578579 0.82 NR1H3 (0.49) ACP1AVPR1BHTR7NR1H2NR1H3
Hydrochloric Acid SCHEMBL6581120 0.81 NR1H3 (0.47) ACP1AVPR1BHTR7NR1H2NR1H3
Hydrochloric Acid SCHEMBL6581321 0.81 NR1H3 (0.48) ACP1AVPR1BHTR7NR1H2NR1H3
Hydrochloric Acid SCHEMBL6580895 0.81 NR1H3 (0.59) ACP1AVPR1BHTR7NR1H2NR1H3
Hydrochloric Acid SCHEMBL6581053 0.81 NR1H3 (0.51) ACP1AVPR1BHTR7NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed