SCHEMBL6587146

SCHEMBL6587146

O=C(Cc1cccc2cnccc12)NCCCc1ccc(C(F)(F)F)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROS1 P08922 1/20 0.53
RPS6KB1 P23443 1/20 0.53
TRPV1 Q8NER1 11/20 0.47
GLS O94925 2/20 0.45
MTNR1A P48039 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583327 0.94 ROS1 (0.55) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL4030518 0.89 ROS1 (0.64) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL6581740 0.83 TRPV1 (0.66) TRPV1
SCHEMBL4023702 0.81 ROS1 (0.61) ROS1RPS6KB1TRPV1GLSMTNR1A
SCHEMBL4030337 0.80 TRPV1 (0.69) ROS1RPS6KB1TRPV1GLSDGAT2
SCHEMBL4019570 0.79 ROS1 (0.69) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL4023632 0.77 ROS1 (0.57) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL6584430 0.77 TRPV1 (0.74) TRPV1
SCHEMBL4023210 0.77 TRPV1 (0.69) ROS1RPS6KB1TRPV1ALDH1A1DGAT2
SCHEMBL4026467 0.76 ROS1 (0.73) ROS1RPS6KB1TRPV1DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478363-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR Abbott Laboratories (US) 2004-11-24 EP claimed
WO-2003070247-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LABORATORIES (US) 2003-08-28 WO claimed