SCHEMBL6584964

SCHEMBL6584964

COc1nccc(N(C)C)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.40
CYP3A4 P08684 4/20 0.40
USP2 O75604 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP2D6 P10635 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
HIF1A Q16665 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CCR1 P32246 1/20 0.38
CCR5 P51681 1/20 0.38
CCR8 P51685 1/20 0.38
RXRA P19793 7/20 0.37
GRIN1 Q05586 7/20 0.37
GRIN2B Q13224 7/20 0.37
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10385800 0.80 CYP1A2 (0.41) CYP1A2CYP3A4USP2KDM4EALDH1A1
SCHEMBL29740313 0.73 NCF1 (0.45) CYP1A2CYP3A4USP2KDM4EALDH1A1
SCHEMBL4268865 0.73 NCF1 (0.45) CYP1A2CYP3A4USP2KDM4EALDH1A1
SCHEMBL1153496 0.71
SCHEMBL30125106 0.71
SCHEMBL1586687 0.71 CYP1A2 (0.47) CYP1A2CYP3A4USP2KDM4EALDH1A1
SCHEMBL12015 0.71 CCR1 (0.41) TDP1CCR1CCR5CCR8RXRA
SCHEMBL29520064 0.71 CCR1 (0.41) TDP1CCR1CCR5CCR8RXRA
SCHEMBL5750346 0.71 CCR1 (0.57) CYP1A2CYP3A4CYP2D6CCR1CCR5
SCHEMBL10568966 0.71 CYP1A2 (0.40) CYP1A2CYP3A4USP2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1455788-A1 1-GLYCINYL-4-AMINOMETHYL-PIPERIDINE DERIVATIVES AS FACTOR XA INHIBITORS ELI LILLY AND COMPANY (US) 2004-09-15 EP disclosed
WO-2003049737-A1 CHEMICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-06-19 WO disclosed