SCHEMBL6584967

SCHEMBL6584967

CC(Oc1cncc(C=Cc2ccncc2)c1)[C@@H]1CCN1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 16/20 0.60
ROCK2 O75116 6/20 0.54
PRKACA P17612 6/20 0.54
ROCK1 Q13464 6/20 0.54
DYRK1A Q13627 6/20 0.54
MAP4K4 O95819 5/20 0.54
PKN2 Q16513 5/20 0.54
CLK4 Q9HAZ1 5/20 0.54
PIM1 P11309 5/20 0.54
CLK2 P49760 4/20 0.54
PRKX P51817 4/20 0.54
PRKG1 Q13976 4/20 0.54
RPS6KB1 P23443 4/20 0.54
DYRK3 O43781 3/20 0.54
CHUK O15111 3/20 0.54
PRKG2 Q13237 3/20 0.54
MKNK2 Q9HBH9 4/20 0.53
STK17A Q9UEE5 4/20 0.53
NTRK3 Q16288 1/20 0.53
CHRNB1 P11230 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8508803 0.94 AKT1 (0.59) AKT1ROCK2PRKACAROCK1DYRK1A
SCHEMBL8508800 0.94 AKT1 (0.59) AKT1ROCK2PRKACAROCK1DYRK1A
SCHEMBL8507932 0.79 AKT1 (0.50) AKT1ROCK2PRKACAROCK1DYRK1A
SCHEMBL8508136 0.78 AKT1 (0.49) AKT1ROCK2ROCK1DYRK1APIM1
SCHEMBL3916101 0.77 AKT1 (0.54) AKT1ROCK2PRKACAROCK1DYRK1A
SCHEMBL3921195 0.77 AKT1 (0.54) AKT1ROCK2PRKACAROCK1DYRK1A
SCHEMBL8508179 0.77 AKT1 (0.54) AKT1ROCK2PRKACAROCK1DYRK1A
SCHEMBL8508178 0.77 AKT1 (0.54) AKT1ROCK2PRKACAROCK1DYRK1A
Hydrochloric Acid SCHEMBL8507893 0.77 AKT1 (0.48) AKT1ROCK2ROCK1DYRK1APIM1
SCHEMBL8507102 0.77 AKT1 (0.39) AKT1ROCK2PRKACAROCK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934308-B1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2004-08-11 EP disclosed