SCHEMBL8508136

SCHEMBL8508136

CC(Oc1cncc(CCc2ccncc2)c1)[C@@H]1CCN1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 5/20 0.49
DAPK3 O43293 1/20 0.49
ROCK2 O75116 1/20 0.49
PRKCG P05129 1/20 0.49
PIM1 P11309 1/20 0.49
RPS6KB1 P23443 1/20 0.49
LIMK1 P53667 1/20 0.49
CDK5 Q00535 1/20 0.49
PRKCD Q05655 1/20 0.49
PAK1 Q13153 1/20 0.49
STK3 Q13188 1/20 0.49
ROCK1 Q13464 1/20 0.49
DYRK1A Q13627 1/20 0.49
CDC42BPA Q5VT25 1/20 0.49
PRKD2 Q9BZL6 1/20 0.49
IRAK4 Q9NWZ3 1/20 0.49
CHRNB2 P17787 3/20 0.47
CHRNB1 P11230 2/20 0.47
CHRNB4 P30926 2/20 0.47
CHRNA3 P32297 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8507893 0.99 AKT1 (0.48) AKT1DAPK3ROCK2PRKCGPIM1
SCHEMBL8508215 0.94 CHRNB2 (0.47) AKT1DAPK3ROCK2PRKCGPIM1
SCHEMBL8508770 0.79 AKT1 (0.41) AKT1DAPK3ROCK2PRKCGPIM1
SCHEMBL6584967 0.78 AKT1 (0.60) AKT1ROCK2PIM1RPS6KB1PRKCD
SCHEMBL8508030 0.77 CHRNA3 (0.35) AKT1DAPK3ROCK2PRKCGPIM1
SCHEMBL6584036 0.76 CHRNB2 (0.69) AKT1DAPK3ROCK2PRKCGPIM1
SCHEMBL6233088 0.76 CHRNB2 (0.40) CHRNB2CHRNB4CHRNA3CHRNA6
SCHEMBL4779704 0.76 CHRNB2 (0.40) CHRNB2CHRNB4CHRNA3CHRNA6
SCHEMBL6236214 0.76 CHRNB2 (0.40) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3
SCHEMBL6234636 0.76 CHRNB2 (0.50) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934308-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 1999-08-11 EP disclosed
WO-1997046554-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1997-12-11 WO disclosed