SCHEMBL6586780

SCHEMBL6586780

CN1CCN(CCCOc2ccc(-c3nc4c(OC(N)=O)cccc4[nH]3)cn2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 4/20 0.52
AURKA O14965 3/20 0.52
PARP1 P09874 5/20 0.50
DRD3 P35462 1/20 0.48
KDR P35968 2/20 0.45
PRKD3 O94806 1/20 0.45
PIM1 P11309 1/20 0.45
SRC P12931 1/20 0.45
FLT4 P35916 1/20 0.45
CLK2 P49760 1/20 0.45
GSK3A P49840 1/20 0.45
DYRK1A Q13627 1/20 0.45
PIM3 Q86V86 1/20 0.45
PRKD2 Q9BZL6 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
STK17A Q9UEE5 1/20 0.45
DHODH Q02127 1/20 0.45
HRH4 Q9H3N8 4/20 0.44
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581381 0.89 PARP1 (0.64) AURKBAURKAPARP1DRD3KDR
SCHEMBL6806452 0.88 AURKB (0.67) AURKBAURKAPARP1KDRPRKD3
SCHEMBL6588600 0.86 AURKB (0.54) AURKBAURKAPARP1DRD3KDR
SCHEMBL6591260 0.86 KDR (0.57) AURKBAURKAPARP1DRD3KDR
SCHEMBL6585555 0.84 AURKB (0.50) AURKBAURKAPARP1DRD3KDR
SCHEMBL6587697 0.84 AURKB (0.44) AURKBAURKAPARP1DRD3KDR
SCHEMBL603789 0.84 DRD3 (0.54) AURKBAURKAPARP1DRD3HRH4
SCHEMBL6588006 0.83 AURKB (0.54) AURKBAURKAPARP1DRD3KDR
SCHEMBL6590927 0.82 AURKB (0.47) AURKBAURKAPARP1DRD3KDR
SCHEMBL7765875 0.82 AURKA (0.77) AURKBAURKAPARP1DRD3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed