SCHEMBL6587643

SCHEMBL6587643

Cc1nc2ccc(-c3nc4cc(N5CCN(C)CC5)ccc4[nH]3)cc2[nH]1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.69
ALDH1A1 P00352 5/20 0.69
TOP1 P11387 3/20 0.69
TOP2A P11388 3/20 0.69
HPGD P15428 1/20 0.69
HSD17B10 Q99714 1/20 0.69
MEN1 O00255 4/20 0.62
KMT2A Q03164 4/20 0.62
MAPT P10636 3/20 0.62
BLM P54132 2/20 0.62
GLA P06280 2/20 0.62
SLCO2B1 O94956 1/20 0.62
RECQL P46063 1/20 0.62
BCL2L1 Q07817 1/20 0.62
SLCO1B3 Q9NPD5 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
SLCO1B1 Q9Y6L6 1/20 0.62
TERT O14746 4/20 0.62
NPC1 O15118 4/20 0.59
RAB9A P51151 4/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587636 0.95 SMN1; SMN2 (0.69) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL18595033 0.94 SMN1; SMN2 (0.77) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL19484928 0.91 ALDH1A1 (0.72) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
Hoechst 33258 SCHEMBL18089342 0.88 ALDH1A1 (0.89) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL23010423 0.87 KDM4E (0.59) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL24299757 0.86 ALDH1A1 (0.65) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL19484925 0.85 ALDH1A1 (0.63) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL8769012 0.84 ALDH1A1 (0.72) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL24299677 0.84 ALDH1A1 (0.62) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD
SCHEMBL13290549 0.84 SMN1; SMN2 (0.60) SMN1; SMN2ALDH1A1TOP1TOP2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9795687-B2 Modularly assembled small molecules for the treatment of myotonic dystrophy type 1 THE SCRIPPS RESEARCH INSTITUTE (US) 2017-10-24 US disclosed
EP-2114896-B1 RADIOPROTECTOR COMPOUNDS AND RELATED METHODS PETER MACCALLUM CANCER INST (AU) 2015-07-22 EP disclosed
US-8796277-B2 Radioprotector compounds and related methods PETER MACCALLUM CANCER INSTITUTE (AU) 2014-08-05 US disclosed
WO-2008074091-A1 RADIOPROTECTOR COMPOUNDS AND RELATED METHODS PETER MACCALLUM CANCER INSTITUTE (AU) 2008-06-26 WO disclosed
EP-0777656-B1 NOVEL DNA-TARGETED ALKYLATING AGENTS AUCKLAND DIVISION CANCER SOC O (NZ) 2004-04-14 EP disclosed
US-5968933-A ANTITUMOR AGENTS AND BINDING DNA FOR MUTAGENESIS AUCKLAND DIVISION CANCER SOCIETY OF NEW ZEALAND INC. (NZ) 1999-10-19 US disclosed
WO-1996006831-A1 NOVEL DNA-TARGETED ALKYLATING AGENTS AUCKLAND DIVISION CANCER SOCIETY OF NEW ZEALAND INC. (NZ) 1996-03-07 WO disclosed