SCHEMBL6589430

SCHEMBL6589430

CC(C)C[C@H](NC(=O)c1cc2cc(OCCN3CCOCC3)ccc2o1)C(=O)NC(C)(C)C(=O)CC(=O)N1CCCCCC1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.55
CTSL P07711 1/20 0.55
CTSB P07858 1/20 0.55
CTSS P25774 1/20 0.55
TAS1R3 Q7RTX0 6/20 0.45
TAS1R1 Q7RTX1 6/20 0.45
PPARG P37231 1/20 0.42
UTS2R Q9UKP6 2/20 0.41
PIN1 Q13526 1/20 0.39
ADAM17 P78536 3/20 0.38
HRH3 Q9Y5N1 1/20 0.38
ACACB O00763 1/20 0.38
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690381 0.77 CTSK (0.75) CTSKCTSLCTSBCTSSTAS1R3
SCHEMBL4690508 0.77 CTSK (0.74) CTSKCTSLCTSBCTSSTAS1R3
SCHEMBL14345772 0.77 CTSK (0.64) CTSKCTSLCTSBCTSSTAS1R3
SCHEMBL5743949 0.76 CTSK (0.57) CTSKCTSLCTSBCTSSTAS1R3
SCHEMBL4765813 0.75 CTSK (0.73) CTSKCTSLCTSBCTSSUTS2R
SCHEMBL5093131 0.75 CTSK (0.73) CTSKCTSLCTSBCTSSTAS1R3
SCHEMBL12632224 0.72 CYP1A2 (0.53) HRH3CYP1A2
SCHEMBL4690446 0.72 CTSK (0.67) CTSKCTSLCTSBCTSSPPARG
SCHEMBL4689513 0.72 CTSK (0.67) CTSKCTSLCTSBCTSS
SCHEMBL15765652 0.71 CTSK (1.00) CTSKCTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed