SCHEMBL6590970

SCHEMBL6590970

C[C@@H](CC(N)=O)CC(=O)NC1CCCN(S(=O)(=O)c2nccs2)CC1=O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 9/20 0.41
CTSL P07711 7/20 0.41
CTSS P25774 7/20 0.41
CTSB P07858 5/20 0.41
CTSV O60911 1/20 0.41
GCK P35557 2/20 0.36
HTT P42858 1/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428085 0.90 CTSK (0.41) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4924362 0.84 CTSK (0.56) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7633224 0.84 CTSK (0.56) CTSKCTSLCTSSCTSBCTSV
SCHEMBL5092610 0.83 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4839973 0.81 CTSK (0.49) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4839956 0.81 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7428075 0.80 CTSK (0.43) CTSKCTSLCTSSCTSBCTSV
SCHEMBL6765207 0.79 CYP3A4 (0.45) CTSKGAAALDH1A1MAPT
SCHEMBL7481625 0.78 CTSK (0.39) CTSKCTSLCTSSCTSBCTSV
SCHEMBL6761962 0.77 POLB (0.46) CTSKCTSLCTSSCTSBCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed