SCHEMBL659267

SCHEMBL659267

Cn1cc(-c2cc3ccnc(N)c3o2)c2ccncc21

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAP3K7 O43318 12/20 0.49
TAB1 Q15750 12/20 0.49
DYRK1A Q13627 2/20 0.48
NFATC1 O95644 1/20 0.48
GSK3B P49841 1/20 0.48
PDPK1 O15530 1/20 0.42
TGFBR1 P36897 1/20 0.42
IKBKE Q14164 1/20 0.42
TBK1 Q9UHD2 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
KDR P35968 2/20 0.42
AURKB Q96GD4 2/20 0.42
TLR8 Q9NR97 2/20 0.40
MAPT P10636 1/20 0.39
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL658287 0.82 MAP3K7 (0.54) MAP3K7TAB1DYRK1ANFATC1GSK3B
SCHEMBL659979 0.79 TLR8 (0.40) MAP3K7TAB1KDRAURKBTLR8
SCHEMBL660235 0.76 LMNA (0.44) MAP3K7TAB1IKBKETBK1TLR8
SCHEMBL659236 0.74 TLR8 (0.40) MAP3K7TAB1KDRAURKBTLR8
SCHEMBL664646 0.74 MAP3K7 (0.64) MAP3K7TAB1KDRAURKBTLR8
SCHEMBL659522 0.71 QPCT (0.39) MAP3K7TAB1TLR8MAPT
SCHEMBL15547185 0.67 DYRK1A (0.77) DYRK1ANFATC1GSK3BPDPK1TGFBR1
SCHEMBL659953 0.67 TLR8 (0.41) MAP3K7TAB1TLR8MAPT
SCHEMBL659131 0.66 MAP3K7 (0.44) MAP3K7TAB1KDRTLR8MAPT
SCHEMBL20385498 0.66 DYRK1A (0.59) DYRK1ANFATC1GSK3BPDPK1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8378104-B2 7-aminofuropyridine derivatives OSI Pharmaceuticals, LLC (US) 2013-02-19 US disclosed
US-20120046267-A1 7-AMINOFUROPYRIDINE DERIVATIVES OSI PHARMACEUTICALS, INC. 2012-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046267-A1 7-AMINOFUROPYRIDINE DERIVATIVES MAP3K5, STK17A, MAPKAPK5 MAP3K7 5/4885TAB1 4/4885DYRK1A 2154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.