SCHEMBL6594758

SCHEMBL6594758

O=C(O)c1cc(O)c2cccc([AsH2])c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
KMT2A Q03164 1/20 0.46
ALOX15 P16050 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
TSHR P16473 2/20 0.41
ACMSD Q8TDX5 1/20 0.41
IGFBP3 P17936 3/20 0.41
RAB9A P51151 2/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.38
GPR35 Q9HC97 2/20 0.37
KDM4A O75164 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
HIF1AN Q9NWT6 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HIF1A Q16665 1/20 0.36
GRIN2D O15399 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xanthurenate SCHEMBL29911018 0.85 KDM4E (0.59) KDM4EKMT2AALOX15TDP1TSHR
Xanthurenate SCHEMBL29394132 0.85 KDM4E (0.59) KDM4EKMT2AALOX15TDP1TSHR
Xanthurenate SCHEMBL379760 0.85 KDM4E (0.59) KDM4EKMT2AALOX15TDP1TSHR
SCHEMBL6080058 0.81 KDM4E (0.46) KDM4EKMT2AALOX15TDP1TSHR
SCHEMBL6080750 0.81 KDM4E (0.46) KDM4EKMT2AALOX15TDP1TSHR
SCHEMBL3333164 0.81 GRM2 (0.48) KDM4EKMT2AALOX15TDP1TSHR
SCHEMBL2909426 0.81 KDM4E (0.49) KDM4EKMT2AALOX15TDP1TSHR
SCHEMBL6079850 0.78 CYP3A4 (0.52) KDM4EKMT2AALOX15ACMSDIGFBP3
SCHEMBL6080552 0.77 KDM4E (0.43) KDM4EKMT2AALOX15TDP1TSHR
SCHEMBL9340049 0.77 KDM4E (0.43) KDM4EKMT2AALOX15TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed