SCHEMBL6594936

SCHEMBL6594936

O=C(O)c1ccc(CN2CCCC2)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
HIF1A Q16665 1/20 0.54
TDP1 Q9NUW8 2/20 0.49
TSHR P16473 1/20 0.49
ALDH1A1 P00352 2/20 0.48
POLB P06746 2/20 0.48
KDM4E B2RXH2 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
HRH3 Q9Y5N1 1/20 0.47
EPHX2 P34913 1/20 0.47
NR1H4 Q96RI1 1/20 0.47
CYP2A13 Q16696 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HSD11B1 P28845 1/20 0.45
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28830570 0.97 CYP2D6 (0.55) IP6K1CYP2D6CYP2C9HIF1ATDP1
SCHEMBL2933311 0.89 ALDH1A1 (0.49) IP6K1TDP1ALDH1A1POLBKDM4E
SCHEMBL4889004 0.87 ALDH1A1 (0.58) IP6K1TDP1TSHRALDH1A1POLB
SCHEMBL12966210 0.83 CXCR4 (0.58) IP6K1ALDH1A1POLB
SCHEMBL13393986 0.82 ALDH1A1 (0.47) TDP1ALDH1A1POLBKDM4EHRH3
SCHEMBL6595744 0.82 ALDH1A1 (0.58) TDP1TSHRALDH1A1POLBKDM4E
SCHEMBL7348167 0.81 GRIN2B (0.54) CYP2D6CYP2C9HIF1AALDH1A1POLB
SCHEMBL20210280 0.81 KDM4E (0.59) CYP2D6CYP2C9HIF1ATDP1ALDH1A1
SCHEMBL7452597 0.81 CYP2D6 (0.54) CYP2D6CYP2C9HIF1ATDP1TSHR
SCHEMBL9456970 0.81 KDM4E (0.55) IP6K1CYP2D6CYP2C9HIF1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-B1 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 2004-12-15 EP disclosed
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed