SCHEMBL6595488

SCHEMBL6595488

CN(C)CCCNC(=O)N1C(=O)/C(=C(/O)c2cccs2)c2cc(Cl)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 1/20 0.44
OPRM1 P35372 3/20 0.42
OPRD1 P41143 3/20 0.42
OPRK1 P41145 3/20 0.42
CCKBR P32239 1/20 0.42
BCHE P06276 1/20 0.39
FLT3 P36888 1/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
DRD2 P14416 2/20 0.37
DRD3 P35462 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
MAPT P10636 1/20 0.36
SNCA P37840 1/20 0.36
BRD4 O60885 1/20 0.35
ASAH1 Q13510 1/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595483 1.00 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
SCHEMBL6595493 1.00 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
SCHEMBL6075746 0.99 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
Hydrochloric Acid SCHEMBL6075397 0.99 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
SCHEMBL6075752 0.99 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
SCHEMBL6075755 0.99 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
Hydrochloric Acid SCHEMBL6075394 0.99 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
Hydrochloric Acid SCHEMBL6075388 0.99 P2RX4 (0.44) P2RX4OPRM1OPRD1OPRK1CCKBR
Hydrochloric Acid SCHEMBL6075712 0.86 OPRM1 (0.40) OPRM1OPRD1OPRK1CCKBRKDM4E
Hydrochloric Acid SCHEMBL6075708 0.86 OPRM1 (0.40) OPRM1OPRD1OPRK1CCKBRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1185526-B1 NOVEL QUATERNARY AMMONIUM DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL USE INST NAT SANTE RECH MED (FR) 2004-09-15 EP disclosed