SCHEMBL6595992

SCHEMBL6595992

COc1cc(N)c(C(=O)Nc2ccccc2)cc1OC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.62
MAPT P10636 4/20 0.62
KDM4E B2RXH2 3/20 0.62
HSD17B10 Q99714 3/20 0.62
HPGD P15428 2/20 0.62
LMNA P02545 2/20 0.62
TP53 P04637 1/20 0.62
ALOX15 P16050 1/20 0.62
TSHR P16473 1/20 0.62
CASP1 P29466 1/20 0.62
CASP7 P55210 1/20 0.62
KCNK3 O14649 2/20 0.57
KCNK9 Q9NPC2 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
KMT2A Q03164 8/20 0.56
NPSR1 Q6W5P4 1/20 0.56
RCE1 Q9Y256 1/20 0.56
MEN1 O00255 6/20 0.55
RAB9A P51151 4/20 0.55
NPC1 O15118 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11088388 0.84 ALDH1A1 (0.55) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL10289035 0.84 NR1H4 (0.56) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL358709 0.83 MAPT (0.54) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL27951004 0.82 ALDH1A1 (0.56) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL17786271 0.81 KDM4E (0.60) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL20388810 0.81 ALDH1A1 (0.55) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL28469086 0.81 BRAF (0.60) MAPTKDM4EHSD17B10TP53CASP1
SCHEMBL7865531 0.81 NPC1 (0.58) MAPTKDM4EHSD17B10TP53CASP1
SCHEMBL733344 0.80 POLB (0.66) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL3177059 0.80 KMT2A (0.53) ALDH1A1MAPTKDM4EHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1143855-C I (ortho)-anthranilamide derivatives as anti-coagulants ���ֹɷݹ�˾ 2004-03-31 CN disclosed
EP-1040108-B1 ORTHO-ANTHRANILAMIDE DERIVATIVES AS ANTI-COAGULANTS SCHERING AG (DE) 2004-02-25 EP disclosed
US-6498185-B1 ENZYME FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. 2002-12-24 US disclosed
US-6380221-B1 FOR THERAPY OF DISEASE-STATES CHARACTERIZED BY THROMBOTIC ACTIVITY BERLEX LABORATORIES, INC. 2002-04-30 US disclosed
CN-1282329-A I (ortho)-anthranilamide derivatives as anti-coagulants SCHERING AG (DE) 2001-01-31 CN disclosed
US-6140351-A FOR TREATING THROMBOSIS BERLEX LABORATORIES, INC. (US) 2000-10-31 US disclosed