SCHEMBL6597703

SCHEMBL6597703

CN(CC(CCN1CCCN(c2nc3ccccc3n2Cc2ccco2)CC1)c1ccccn1)C(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 10/20 0.41
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
TACR1 P25103 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
OPRD1 P41143 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6597773 0.92 TACR2 (0.46) TACR2MEN1ALDH1A1GAAMAPT
SCHEMBL6599750 0.91 HRH1 (0.42) TACR2MEN1ALDH1A1GAAMAPT
SCHEMBL6597481 0.90 TACR2 (0.44) TACR2MEN1ALDH1A1GAAMAPT
SCHEMBL6594816 0.90 TACR2 (0.41) TACR2HTTTACR1SMN1; SMN2NPSR1
SCHEMBL6598719 0.89 TACR2 (0.42) TACR2MEN1ALDH1A1GAAMAPT
SCHEMBL6597572 0.89 TACR2 (0.41) TACR2
SCHEMBL6596324 0.88 TACR2 (0.45) TACR2MEN1ALDH1A1GAAMAPT
SCHEMBL6597730 0.88 TACR2 (0.49) TACR2TACR1
SCHEMBL6594419 0.88 TACR2 (0.48) TACR2TACR1
SCHEMBL6600342 0.87 LMNA (0.45) TACR2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888338-B1 NOVEL SUBSTITUTED N-METHYL-N-(4-(4-(1H-BENZIMIDAZOL-2-YL) 1,4]DIAZEPAN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES AVENTIS PHARMA INC (US) 2004-11-17 EP disclosed