SCHEMBL6598211

SCHEMBL6598211

CS(=O)(=O)c1ccc(C2=C(c3ccccc3)C(=O)OC2[SeH])cc1

nearest known ligand 0.71

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 0.71
PTGS1 P23219 10/20 0.52
ABCB11 O95342 1/20 0.52
ALDH1A1 P00352 1/20 0.52
MT-CO2 P00403 1/20 0.52
HTR1A P08908 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
MC4R P32245 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21675747 0.84 PTGS2 (0.72) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL6672818 0.84 PTGS2 (0.72) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL21675748 0.83 PTGS2 (0.71) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
5-Hydroxy Rofecoxib SCHEMBL6331980 0.83 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL17917317 0.81 PTGS2 (0.67) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7958864 0.80 PTGS2 (0.70) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL6676482 0.78 PTGS2 (0.63) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL6676479 0.77 PTGS2 (0.62) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL8423806 0.75 PTGS2 (0.69) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL7567581 0.75 PTGS2 (0.59) PTGS2PTGS1ABCB11ALDH1A1MT-CO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414526-A2 ANTIANGIOGENIC COMBINATION THERAPY FOR THE TREATMENT OF CANCER Pharmacia Corporation (US) 2004-05-06 EP disclosed
WO-2002085459-A2 ANTIANGIOGENIC COMBINATION THERAPY FOR THE TREATMENT OF CANCER PHARMACIA CORPORATION (US) 2002-10-31 WO disclosed
EP-1140179-A2 USE OF A CYCLOOXYGENASE 2 INHIBITOR AND AN INTEGRIN ANTAGONIST AS A COMBINATION THERAPY IN THE TREATMENT OF NEOPLASIA G.D. SEARLE & CO. (US) 2001-10-10 EP disclosed
WO-2000038786-A2 USE OF CYCLOOXYGENASE 2 INHIBITOR AND AN INTEGRIN ANTAGONIST AS A COMBINATION THERAPY IN THE TREATMENT OF NEOPLASIA G.D. SEARLE & CO. (US) 2000-07-06 WO disclosed