SCHEMBL6598792

SCHEMBL6598792

O=C(O)c1c2c(cc3nc(-c4ccccc4)c(CN4CCC(N5CCCCC5)CC4)cc13)OCO2

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 5/20 0.49
TACR3 P29371 5/20 0.49
TRPV4 Q9HBA0 15/20 0.48
OPRM1 P35372 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6394399 0.87 TACR2 (0.57) TACR2TACR3TRPV4OPRM1
Hydrochloric Acid SCHEMBL6399854 0.86 TACR2 (0.57) TACR2TACR3TRPV4OPRM1
SCHEMBL5203685 0.82 TACR2 (0.57) TACR2TACR3TRPV4OPRM1
SCHEMBL5202474 0.81 TACR3 (0.59) TACR2TACR3TRPV4OPRM1
SCHEMBL2373330 0.76 TRPV4 (0.72) TACR2TACR3TRPV4OPRM1
Hydrochloric Acid SCHEMBL5733490 0.75 TRPV4 (0.71) TACR2TACR3TRPV4OPRM1
SCHEMBL5945353 0.75 TRPV4 (0.63) TACR2TACR3TRPV4OPRM1
SCHEMBL5945435 0.75 TRPV4 (0.59) TACR2TACR3TRPV4OPRM1
SCHEMBL6393346 0.75 TRPV4 (0.58) TACR2TACR3TRPV4OPRM1
SCHEMBL5945404 0.74 TRPV4 (0.62) TACR2TACR3TRPV4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377555-A1 NOVEL COMPOUNDS GlaxoSmithKline S.p.A. (IT) 2004-01-07 EP disclosed
WO-2002083645-A1 NOVEL COMPOUNDS GLAXOSMITHKLINE S.P.A. (IT) 2002-10-24 WO disclosed