SCHEMBL6600824

SCHEMBL6600824

Cc1cccc2oc(N3CCN4CCC3CC4)nc12

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 5/20 0.64
CHRNA7 P36544 4/20 0.64
KCNH2 Q12809 3/20 0.60
CHRM4 P08173 1/20 0.60
CHRM5 P08912 1/20 0.60
CHRM1 P11229 1/20 0.60
CHRM3 P20309 1/20 0.60
CHRNB4 P30926 1/20 0.60
CHRNA3 P32297 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5154912 0.99 HTR3A (0.62) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL4704458 0.80 HTR3A (0.58) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL4701401 0.79 HTR3A (0.64) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL373021 0.78 HTR3A (1.00) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL4699052 0.75 HTR3A (1.00) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL4699915 0.75 HTR3A (0.69) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL4700653 0.75 HTR3A (0.69) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL1459339 0.75 HTR3A (1.00) HTR3ACHRNA7KCNH2CHRM4CHRM5
Hydrochloric Acid SCHEMBL15663033 0.74 HTR3A (0.97) HTR3ACHRNA7KCNH2CHRM4CHRM5
SCHEMBL5248370 0.74 HTR3A (0.77) HTR3ACHRNA7KCNH2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289988-B1 1,4-DIAZABICYCLO 3.2.2]NONABENZOXAZOLE, -BENZOTHIAZOLE AND BENZIMIDAZOLE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI SYNTHELABO (FR) 2004-05-19 EP disclosed