SCHEMBL6601533

SCHEMBL6601533

COc1ccccc1CCn1c(CO[Si](C)(C)C(C)(C)C)cnc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.42
CYP3A4 P08684 7/20 0.42
CYP2C9 P11712 7/20 0.42
TSHR P16473 7/20 0.42
CYP2C19 P33261 7/20 0.42
USP2 O75604 5/20 0.42
CYP2D6 P10635 4/20 0.42
ALDH1A1 P00352 4/20 0.42
CLK4 Q9HAZ1 2/20 0.42
LMNA P02545 2/20 0.42
HIF1A Q16665 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
KCNH2 Q12809 2/20 0.40
HRH3 Q9Y5N1 1/20 0.40
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDM4E B2RXH2 2/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601369 0.80 SIGMAR1 (0.48) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
Hydrochloric Acid SCHEMBL6602964 0.79 KCNH2 (0.49) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6602683 0.79 SIGMAR1 (0.42) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL1247733 0.72 TAAR1 (0.50) ALDH1A1LMNASIGMAR1KCNH2HRH3
SCHEMBL30416922 0.70 TAAR1 (0.47) ALDH1A1LMNASIGMAR1KCNH2HRH3
SCHEMBL30416478 0.70 TAAR1 (0.47) ALDH1A1LMNASIGMAR1KCNH2HRH3
SCHEMBL6601527 0.70 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6601984 0.66 KDM4E (0.47) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6601534 0.65 CYP2C19 (0.30) CYP2C19
SCHEMBL20189141 0.65 IDO1 (0.44) ALDH1A1LMNAKDM4EIDO1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1169320-B1 FARNESYL TRANSFERASE INHIBITORS HAVING A PYRROLE STRUCTURE AND PROCESS FOR PREPARATION THEREOF LG CHEM INVESTMENT LTD (KR) 2004-09-22 EP disclosed
US-6511978-B1 For treating cancer, restenosis, atherosclerosis or viral infections LG LIFE SCIENCES, LTD. (KR) 2003-01-28 US disclosed